藥物與人體作用之機制，藥物之化學構造及設計原理。

1. drug names and chemical structures 2. drug mechanisms and uses 3. drug stereochemistry and conformations 4. drug pharmacophore and pharmacology 5. structure-activity relationship (SAR): drug-enzyme (or receptor) interactions and complex cocrystal structures 6. drug design, discovery, synthesis (case study)

1. Foye’s Principles of Medicinal Chemistry 6th ed., 2007 William O. Foye, Editor: Lemke and Williams
2. Essentials of Foye’s Principles of Medicinal Chemistry, 2016, Editor: T. L. Lemke, S. W. Zito, V. F. Roche, D. A. Willaims